Darunavir (Ethanolate)

CAS: 635728-49-3

Category: Pharmaceutical Intermediates

PurityReagent Grade ≥98%, High-Purity Grade ≥99%, Pharmaceutical Grade ≥99.5%
Molecular FormulaC29H43N3O8S
Molecular Weight593.73
Appearancewhite to off-white crystalline powder
Packaging25 kg/fiber drum, 1 kg/aluminum foil bag.
Testing IndicatorsAppearance — Visual inspection; Identification — IR, Chiral HPLC; Purity — Gradient RP-HPLC; Enantiomeric purity — Chiral HPLC; Ethanol — HS-GC; Heavy metals — ICP-MS; Moisture — Karl Fischer titration; Microbial limits — Membrane filtration; Protease sulfonamides — LC-MS.
Storage NotesStored in a cool, dry, and well-ventilated place at room temperature in a tightly closed container, protected from light and moisture.
Lead Time days
Used as a HIV protease inhibitor intermediate in the synthesis of oral boosted antiretroviral agents for treatment-experienced HIV-1 infection.