Argatroban

CAS: 74863-84-6

Category: Organic Pharmaceutical Intermediates

PurityResearch/API grade typically ≥98% purity (HPLC), with defined limits for related substances, residua
Molecular FormulaC23H36N6O5S
Molecular Weight508.63
AppearanceWhite to off-white solid (crystalline or amorphous powder)
PackagingResearch scale: 1 mg–100 mg glass vials or small bottles; API/bulk scale: multi-gram to multi-kilogram sealed bottles or drums with moisture and light protection, intended for pharmaceutical and research use
Testing IndicatorsAppearance — visual inspection (color and form); Assay and related substances — HPLC; Identification — ¹H/¹³C NMR, FTIR, and MS, including HPLC retention versus reference; Water content — Karl Fischer titration; Residual solvents — GC; Specific rotation — polarimetry where specified by quality standards.
Storage NotesStore in a tightly closed container in a cool, dry place (typically 2–8 °C or below) protected from light and moisture. Avoid prolonged exposure to elevated temperature and humidity, and keep away from strong oxidizing agents and incompatible chemicals. For solutions, follow specified stability and storage conditions.
Lead Time10 days
Synthetic direct thrombin inhibitor used as a non-heparin anticoagulant and pharmaceutical active/intermediate. Applied clinically (in appropriate dosage forms) for the prevention and treatment of thrombosis, especially in patients with heparin-induced thrombocytopenia (HIT), and used as a research tool in thrombosis and coagulation studies.